Претраживање
Приказ резултата 1-10 од 11
Second Generation Steroidal 4-Aminoquinolines Are Potent, Dual-Target Inhibitors of the Botulinum Neurotoxin Serotype A Metalloprotease and P. falciparum Malaria
(American Chemical Society (ACS), 2014)
Significantly more potent second generation 4-amino-7-chloroquinoline (4,7-ACQ) based inhibitors of the botulinum neurotoxin serotype A (BoNT/A) light chain were synthesized. Introducing an amino group at the C(3) position ...
A Chemotype That Inhibits Three Unrelated Pathogenic Targets: The Botulinum Neurotoxin Serotype A Light Chain, P. falciparum Malaria, and the Ebola Filovirus
(American Chemical Society (ACS), 2011)
A 1,7-bis(alkylamino)diazachrysene-based small molecule was previously identified as an inhibitor of the botulinum neurotoxin serotype A light chain metalloprotease. Subsequently, a variety of derivatives of this chemotype ...
alpha-Glucosidase inhibitory activity and cytotoxic effects of some cyclic urea and carbamate derivatives
(Taylor & Francis Ltd, Abingdon, 2017)
The inhibitory activities of selected cyclic urea and carbamate derivatives (1-13) toward alpha-glucosidase (alpha-Gls) in in vitro assay were examined in this study. All examined compounds showed higher inhibitory activity ...
Five primary sources of organic aerosols in the urban atmosphere of Belgrade (Serbia)
(Elsevier, 2016)
Biomass burning and primary biological aerosol particles (PBAPs) represent important primary sources of organic compounds in the atmosphere. These particles and compounds are able to affect climate and human health. In the ...
Evaluation of potentially toxic element contamination in the riparian zone of the River Sava
(Elsevier, 2019)
Contaminated sediments transported onto the river terrace during high water events can contribute significant quantities of potentially toxic elements to riparian soils. Seven trace elements (As, Cd, Cr, Cu, Ni, Pb and Zn) ...
Significance of diarylheptanoids for chemotaxonomical distinguishing between Alnus glutinosa and Alnus incana
(Walter De Gruyter, 2018)
Diarylheptanoids are a group of secondary metabolites widely distributed in the Betulaceae family and characteristic for Alnus species. In this study, the chemotaxonomic power of diarylheptanoids, such as hirsutanonol-5- ...
RuxTi1-xO2 as the support for Pt nanoparticles: Electrocatalysis of methanol oxidation
(Elsevier, 2015)
Two binary Ru-Ti oxides, Rum Ti0.9O2 and Ru0.7Ti0.3O2, were synthesized by the sol-gel method and used as an electrocatalyst support. The system was characterized by XRD, EDS, TEM and cyclic voltammetry. The Rum Ti0.9O2 ...
Conformational stability of digestion-resistant peptides of peanut conglutins reveals the molecular basis of their allergenicity
(Nature Publishing Group, London, 2016)
Conglutins represent the major peanut allergens and are renowned for their resistance to gastrointestinal digestion. Our aim was to characterize the digestion-resistant peptides (DRPs) of conglutins by biochemical and ...
Understanding the Effect of Energy Density and Formulation Factors on the Printability and Characteristics of SLS Irbesartan Tablets-Application of the Decision Tree Model
(MDPI, 2021)
Selective laser sintering (SLS) is a rapid prototyping technique for the production of three-dimensional objects through selectively sintering powder-based layer materials. The aim of the study was to investigate the effect ...
Immobilization of biocatalysts for enzymatic polymerizations: Possibilities, advantages, applications
(Elsevier Sci Ltd, Oxford, 2012)
Biotechnology also holds tremendous opportunities for realizing functional polymeric materials. Biocatalytic pathways to polymeric materials are an emerging research area with not only enormous scientific and technological ...