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Приказ резултата 1-10 од 19
7, 8, 15, 16-Tetraoxa-dispiro [5. 2. 5. 2]hexadecane-3-carboxylic acid derivatives and their antimalarial activity / Antimalarijska aktivnost derivata 7,8,15,16-tetraoksa-dispiro5.2.5.2heksadekan-3-karboksilne kiseline
(Serbian Chemical Society, 2004)
Several C2 symmetrical mixed tetraoxanes were prepared starting from a gemdihydroperoxide and a ketone. The obtained tetraoxanes showed pronounced antimalarial activity against P. falciparum chloroquine resistant W2 and ...
Stereoselective synthesis of α-hydroxy-β-amino acids: The chiral pool approach / Stereoselektivne sinteze α-hidroksi-β-aminokiselina iz prirodnih hiralnih prekursora
(Serbian Chemical Society, 2004)
A method for the stereoselective homologation of -amino acids into syn-α-hydroxy-β-amino acids is described, based on the conversion of stereoisomeric cyanohydrins into trans-oxazolines. The synthetic potential of the ...
Effect of MnSOD (E. coli) on the relaxation caused by sodium nitroprusside on isolated rat renal artery / Efekat MnSOD (E. coli) Na relaksaciju izolovane renalne arterije pacova izazvanu natrijum-nitro-prusidom
(Serbian Chemical Society, 2004)
In this study themolecular foundation of nitric oxide induced relaxation of arteries, with or without endothelium, of normotensive and spontanously hypertensive ratswas re-examined. With this purpose in mind, the effects ...
Modeling of adsorber/desorber/catalytic reactor system for ethylene oxide removal / Modelovanje sistema adsorber/desorber/katalitički reaktor za uklanjanje etilen oksida
(Serbian Chemical Society, 2004)
The removal of ethylene oxide (EtO) in a combined system adsorber desorber/catalytic reactor has been investigated. The combined system was a modified draft tube spouted bed reactor loaded with Pt/Al2O3 catalyst. The annular ...
Noble metal binding on macroporous poly(GMA-co-EGDMA) modified with ethylenediamine / Vezivanje plemenitih metala za makroporozni poli(GMA-co-EGDMA)kopolimer modifikovan sa etilendiaminom
(Serbian Chemical Society, 2004)
Macroporous crosslinked poly(glycidyl methacrylate-co-ethylene glycol dimethacrylate), p(GME), was synthesized by suspension copolymerization and modified by reaction of the pendant epoxy groups with ethylenediamine. The ...
The synthesis and pharmacological evaluation of (+/-)-2,3-seco-fentanyl analogues / Sinteza i farmakološko ispitivanje (±)-2,3-seco-analoga fentanila
(Serbian Chemical Soc, Belgrade, 2004)
An efficient, five-step synthetic approach to various acyclic 1,3-diamines has been developed and applied to the preparation of a novel class of open-chained fentanyl analogues. The acyclic derivatives 5.1-5.5 (all new ...
The synthesis and preliminary pharmacological evaluation of the racemic cis and trans 3-alkylfentanyl analogues / Sinteza i preliminarni farmakološki testovi recemskih cis i trans 3-alkilanaloga fentanila
(Serbian Chemical Soc, Belgrade, 2004)
A general five step method for the synthesis of 3-alkylfentanyl analogues (i.e. cis and trans 3-alkyl-4-anilidopiperidines 6.1-6.6) has been developed, The starting N-phenethyl-4-piperidone 1 was first converted into the ...
Antifungal activity of davanone-type sesquiterpenes from Artemisia lobelii var. conescens / Antifungalna aktivnost terpenoida davanonskog tipa izolovanih iz Artemisia lobelii Var. canescens
(Serbian Chemical Soc, Belgrade, 2004)
Five tetrahydrofuran sesquiterpenes, so-called davanones, and coumarin umbelliferone isolated from Artemisia lobelii All. var. canescens (DC.) Briqu, were tested for antifungal activity. All the compounds inhibited the ...
Synthesis of 5-azaandrostane-3β,17β-diol protected at the 17β-hydroxyl group
(Serbian Chemical Society, 2004)
In the present paper, the preparation of 3β-hydroxy-17β-dimethyl- tert-butylsilyloxy-5-azaandrostane (15) in fourteen steps is described. B-nor-17-oxoandrost-5-en-3β-yl acetate (1) 1,2 was used as the starting material, ...
Protein covalent modification of biologically active quinones / Kovalentne modifikacije proteina biološki aktivnim hinonima
(Serbian Chemical Society, 2004)
The avarone/avarol quinone/hydroquinone couple shows considerable antitumor activity. In this work, covalent modification of β-lactoglobulin by avarone and its derivatives as well as by the synthetic steroidal quinone ...