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Structure-activity relationship study of steroidal 1,2,4,5-tetraoxane animalarials using computational procedures / QSAR izučavanje steroidnih 1,2,4,5-tetraoksanskih antimalarika računarskim modelovanjem
(Serbian Chemical Society, 2005)
A three-dimensional QSAR pharmacophore model for antimalarial activity of steroidal 1,2,4,5-tetraoxanes was developed from a set of 17 substituted antimalarial derivatives out of 27 analogues that exhibited remarkable in ...
alpha-Glucosidase inhibitory activity and cytotoxic effects of some cyclic urea and carbamate derivatives
(Taylor & Francis Ltd, Abingdon, 2017)
The inhibitory activities of selected cyclic urea and carbamate derivatives (1-13) toward alpha-glucosidase (alpha-Gls) in in vitro assay were examined in this study. All examined compounds showed higher inhibitory activity ...
A QSAR study of acute toxicity of N-substituted fluoroacetamides to rats
(Oxford : Pergamon-Elsevier Science Ltd, 2006)
Acute toxicity in vivo toward rats, of nineteen N-alkyl and N-cycloalkyl fluorocetamides [F-CH2-C(O)-NH-R] was correlated with their structure-dependent properties. Used descriptors are: molecular weights (M-w) and heat ...
Substitued (E)-β-(benzoyl)acrylic acids suppressed survival of neoplastic human HeLa cells / Umanjeno preživljavanje neoplastičkih humanih HeLa ćelija supstituisanim (E)-b-(benzoil) akrilnim kiselinama
(Belgrade : Serbian Chemical Society, 1999)
The bacteriostatic activity of some of alkyl substituted (E)-β-(benzoyl)acrylic acids was shown earlier. The aim of this study was to investigate the antiproliferative action of 19 alkyl-, or halogeno-, or methoxy-, or ...
Antiproliferative activity of β-hydroxy- β-arylalkanoic acids
(MDPI, 2007)
Article describes the synthesis of fifteen β-hydroxy- β-arylalkanoic acids by Reformatsky reaction using the 1-ethoxyethyl-2- bromoalkanoates, aromatic or cycloalkyl ketones or aromatic aldehydes. The short survey of ...
Environmental hazard assessment of the newly synthetized substances as corrosion inhibitors with potential environment friendly industrial application as anticorrosive agent in paints and coatings for the river and sea vessels by using QSAR models for prediction of their physico-chemical and eco- toxicological properties
(Association of Chemistry and the Environment, 2022)
Due to global environmental policy goals to reduce marine and ocean pollutions, there is a global need to finding greener solutions for industrial chemicals design in line with principle of the green chemistry. Therefore, ...