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Synthesis and pharmacological evaluation of novel cis and trans 3‑substituted anilidopiperidines
(Springer Nature, 2020)
Background 4-Anilidopiperidine class of synthetic opioid analgesics, with it’s representative fentanyl, are by far the most potent and clinically significant for the treatment of the severe chronic and surgical pain. ...
Experimental examination and thermodynamic description of the ternary Bi-Ge-Ga,Zn systems
(Elsevier, 2020)
Due to the wide application of systems based on germanium ternary Bi-Ga-Ge and Bi-Ge-Zn systems were experimentally tested in this study. Used experimental techniques were scanning electron microscope with energy dispersive ...
Chemo- and biocatalytic esterification of marchantin A and cytotoxic activity of ester derivatives
(Elsevier, 2020)
Chemical and biocatalytic synthesis of seven previously undescribed marchantin A ester derivatives has been presented. Chemical synthesis afforded three peresterified bisbibenzyl products (TE1-TE3), while enzymatic method, ...
The time response of plasmonic sensors due to binary adsorption: analytical versus numerical modeling
(Springer Nature, 2020)
In order to allow for multiscale modeling of complex systems we focus on various approaches to modeling binary adsorption. We consider multiple methods of modeling the temporal response of general plasmonic sensors. We ...
Formulation and characterization of novel liposomes containing histidine for encapsulation of a poorly soluble vitamin
(Elsevier, 2020)
In this study, development of folic acid-loaded liposomes using a basic amino acid, histidine as a solubilizing agent for folic acid was presented, which tackled the poor solubility of this vitamin. The effect of the ...
Self-Assembly and Biorecognition of a Spirohydantoin Derived from α-Tetralone: Interplay between Chirality and Intermolecular Interactions
(John Wiley and Sons Inc., 2020)
A racemic spirohydantoin derivative with two aromatic substituents, a tetralin and a 4-methoxybenzyl unit, was synthesized and its crystal structure was determined. To define the relationship between molecular stereochemistry ...
Bisaurones-enzymatic production and biological evaluation
(Royal Society of Chemistry, 2020)
The Trametes versicolor laccase catalyzed oxidation of chalcone butein afforded four dimers of aurone sulfuretin (i.e. two regioisomeric pairs of diasteromers, 1-4) as the major products. The formation of the dimers was ...
Increased yield of enzymatic synthesis by chromatographic selection of different N-glycoforms of yeast invertase
(Wiley, 2020)
Invertases are glycosidases applied for synthesis of alkyl glycosides that are important and effective surfactants. Stability of invertases in the environment with increased content of organic solvent is crucial for increase ...
Multi-disciplinary Shape Optimization of Missile Fin Configuration Subject to Aerodynamic Heating
(American Institute of Aeronautics and Astronautics, 2020)
The main goal of this paper is to expand previously conducted study and consequently to upgrade the proposed multimodular numerical framework developed for fluid–structure interaction simulation (FSI) and multidisciplinary ...
Modulating Excited Charge-Transfer States of G‑Quartet Self- Assemblies by Earth Alkaline Cations and Hydration
(American Chemical Society (ACS), 2020)
Guanine self-assemblies are promising supramolecularplatforms for optoelectronic applications. The study (Hua et al., J. Phys. Chem. C 2012, 116, 14,682−14,689) reported that alkaline cations cannot modulate the electronic ...