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Synthesis and dopaminergic properteis of 3- and 4-substituted 1-{-[5-(1H-benzimidazole-2-thione)]ethyl}piperidines and related compounds
(Wiley, 1997)
With an aim of creating new, high affinity dopaminergic ligands, six different 3- and 4-substituted 1-{2-[5-(1H-benzimidazole-2-thione)]ethyl}piperidines and nine related heterocyclic congeners were synthesized and evaluated ...
Electron‐impact induced decomposition of some 3‐alkyl‐5‐substituted‐6‐methyl uracils
(John Wiley & Sons, 1995)
Mass spectrometry was used to study the main fragmentation routes of some 3‐alkyl‐5‐substituted‐6‐methyl uracils. Differences in fragmentation were caused by changes in the structure of the alkyl group in position 3 of the ...
Modeling of drawing thin glass sheet from a preform / Model izvlačenja tankih staklenih traka iz predoblika
(Serbian Chemical Society, 1998)
A one-dimensional model of thin glass sheet drawing has been developed. This model includes momentum, heat and mass balance equations. The density, viscosity and specific heat of the glass were calculated as functions of ...
Photochemically induced mercuric oxide - iodine oxidation of some unsaturated steroid compounds
(Pergamon, 1994)
Photochemically induced HgO/I2 oxidation of cholest-5-en-3α-ol (6) and cholest-5-en-3β-ol (7) afforded (Scheme 3) products arising from the corresponding alkoxy radicals (12, 13 and 14a,b) and from attack of the I2O ...
New substituted 2-methylthiomethyl- and 2-methylsulphinylmethylenebenz- imidazoles with D 2 /5-HT(1A) activity
(Govi-Verlag Pharmazeutischer Verlag GmbH, 1998)
Several 2-methylthiomethylbenzimidazoles (3a-e) and the corresponding sulphinyl derivatives 4a-e were synthesized and evaluated measuring their in vitro binding affinity at the D 1 and D 2 dopamine (source: synaptosomal ...
Synthesis and dopaminergic features of six novel 3-arylpiperidines
(Bollettino Chimico Farmaceutico, 1998)
Four substituted 3-aryl-1-{2-[5-(1H-benzimidazole)]ethyl}piperidines and two 3-aryl-1-{2-[6-(1,4-dihydroxyquinoxaline-2,3-dione)]ethyl} piperidines were synthesized, characterized and evaluated for in vitro binding affinity ...
Synthesis of several substituted phenylpiperazines behaving as mixed D2/5HT(1A) ligands
(Blackwell Publishing Ltd, 1997)
Twenty-two different compounds have been synthesized with the aim of creating new, mixed D2/5HT(1A) ligands. For this purpose l-substituted phenylpiperazines attached by the N-4 nitrogen to dopaminergic pharmacophores of ...
Novel 5-[2-(N,N-di-n-propylamino)-ethyl]benzimidazole-derived high affinity dopaminergic ligands
(Govi-Verlag Pharmazeutischer Verlag GmbH, 1996)
Derivatives of a noncatechol dopamine (DA) bioisostere 5-[2-(N,N-di-n-propylamino)ethyl]-benzimidazole (15) were synthesized and checked for affinity towards D-1 and D-2 DA receptors (DAR). Ten compounds were obtained by ...
Free radical ring expansion and subsequent reactions of intermediary carbon radicals
(Serbian Chemical Society, 1996)
Alkyl radicals, derived from ethyl 1-(bromoalkyl)-2-oxocyclo-alkanecarboxylates or from the corresponding thiohydroxamic esters, undergo a ring expansion reaction and subsequent intermoleculaar addition/elimination reactions. ...
Corrosion protection of aluminium by a cataphoretic epoxy coating
(Elsevier, 1999)
The corrosion behavior and thermal stability of epoxy coating electrodeposited on aluminium have been investigated during exposure to
3% NaCl. Electrochemical impedance spectroscopy (EIS), gravimetric liquid sorption ...