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Leucine aminopeptidase from Streptomyces hygroscopicus is controlled by a low molecular weight inhibitor
(Society of Fermentation and Bioengineering, 2002)
In culture filtrate of Streptomyces hygroscopicus a producer of polyketide antibiotics, a leucine aminopeptidase and its autogenous inhibitor were detected. The leucine aminopeptidase was purified 4573-fold with yield of ...
Synthesis, dopamine D-2 receptor binding studies and docking analysis of 5-[3-(4-arylpiperazin-1-yl)propyl]-1H-benzimidazole, 5-[2-(4-arylpiperazin-1-yl)ethoxy]-1H-benzimidazole and their analogs
(Editions Scientifiques Medicales Elsevier, Paris, 2005)
5-[3-(4-Arylpiperazin-1-yl)propyl]-1H-benzimidazoles and 5-[2-(4-aryipiperazin-1-yl)ethoxy]-1H-benzimidazoles were synthesized and their affinity for the D-1, D-2 and 5-HT1A, receptors examined. They expressed a rather ...
1-Cinnamyl-4-(2-methoxyphenyl)piperazines: Synthesis, binding properties, and docking to dopamine (D2) and serotonin (5-HT1A) receptors
(Wiley-V C H Verlag Gmbh, Weinheim, 2007)
Clinical properties of atypical antipsychotics are based on their interaction with D2 dopamine receptor and serotonin 5-HT1A and 5-HT2A receptors. As a part of our research program on new antipsychotics, we synthesized ...
Synthesis, binding properties and receptor docking of 4-halo-6-[2-(4-arylpiperazin-1-yl)ethyl]-1H-benzimidazoles, mixed ligands of D2 and 5-HT1A receptors
(Elsevier France-Editions Scientifiques Medicales Elsevier, Issy-Les-Moulineaux, 2008)
In this publication we are describing synthesis, binding properties, and receptor docking of 4-halo-6-[2-(4-arylpiperazin-1-yl)ethyl]-1H-benzimidazoles, a new compounds with potential antipsychotics properties. Affinity ...
Phenolics, lignin content and peroxidase activity in Picea omorika lines
(Biologia Plantarum, 2006)
We analyzed low molecular mass phenolics, lignin content and both soluble and cell wall bound peroxidase activity in the needles of three Picea omorika (Pancic) Purkyne lines grown in the generative seed orchard. The highest ...
Relationships between structure, retention and biological activity of some Schiff base ligands and their complexes
(Biomedical Chromatography, 2008)
The lipophilicity of a series of Schiff base ligands and their complexes with nickel(II) and copper(II) has been determined by reversed-phase thin-layer chromatography using binary dioxane-water mobile phase. Chelate ligands ...
Effects of O2+ ions beam irradiation on crystal structure of rare earth sesquioxides
(Elsevier, 2009)
We report the results of ion irradiation influence on rare earth sesquioxides structure, which are materials of practical importance as a radiation resistant ceramics in nuclear applications. Y2O3, Gd2O3 and Er2O3 sesquioxides ...
Introduction of a methyl group in alpha- or beta-position of 1-heteroarylethyl-4-phenyl-piperazines affects their dopaminergic/serotonergic properties
(Wiley-VCH Verlag Gmbh, Weinheim, 2001)
1-(2-Heteroarylalkyl)-4-phenylpiperazines containing methyl group in either the alpha- or the beta-position of the side alkyl chain were synthesized as racemic mixtures. They were evaluated for in vitro binding affinity ...
Role of complexes formation between drugs and penetration enhancers in transdermal delivery
(Elsevier, 2008)
The use of chemical penetration enhancers (CPE) is growing due to their ability to improve drug delivery through the skin. A possible mechanism of penetration enhancement could involve the complex formation between drug ...
Pulse and direct current plating of Ni-W alloys from ammonia-citrate electrolyte
(Elsevier, 2006)
The effect of the potential of deposition and electrode rotation rate on current efficiency and partial current density of nickel deposition from ammonia-citrate electrolyte with and without tungstate ions was investigated. ...