Bihelović, Filip

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Authority KeyName Variants
orcid::0000-0002-7654-3189
  • Bihelović, Filip (10)
Projects

Author's Bibliography

Development of iminosugar-based glycosidase inhibitors as drug candidates for SARS-CoV-2 virus via molecular modelling and in vitro studies

Ferjančić, Zorana; Bihelović, Filip; Vulović, Bojan; Matović, Radomir; Trmčić, Milena; Janković, Aleksandar; Pavlović, Miloš; Đurković, Filip T.; Prodanović, Radivoje; Đurđević Đelmaš, Aleksandra; Kaličanin, Nevena; Zlatović, Mario; Sladić, Dušan; Vallet, Thomas; Vignuzzi, Marco; Saičić, Radomir N.

(Taylor and Francis Group, 2024)

TY  - JOUR
AU  - Ferjančić, Zorana
AU  - Bihelović, Filip
AU  - Vulović, Bojan
AU  - Matović, Radomir
AU  - Trmčić, Milena
AU  - Janković, Aleksandar
AU  - Pavlović, Miloš
AU  - Đurković, Filip T.
AU  - Prodanović, Radivoje
AU  - Đurđević Đelmaš, Aleksandra
AU  - Kaličanin, Nevena
AU  - Zlatović, Mario
AU  - Sladić, Dušan
AU  - Vallet, Thomas
AU  - Vignuzzi, Marco
AU  - Saičić, Radomir N.
PY  - 2024
UR  - https://cer.ihtm.bg.ac.rs/handle/123456789/7585
AB  - We developed new iminosugar-based glycosidase inhibitors against SARS-CoV-2. Known drugs (miglustat, migalastat, miglitol, and swainsonine) were chosen as lead compounds to develop three classes of glycosidase inhibitors (α-glucosidase, α-galactosidase, and mannosidase). Molecular modelling of the lead compounds, synthesis of the compounds with the highest docking scores, enzyme inhibition tests, and in vitro antiviral assays afforded rationally designed inhibitors. Two highly active α-glucosidase inhibitors were discovered, where one of them is the most potent iminosugar-based anti-SARS-CoV-2 agent to date (EC90 = 1.94 µM in A549-ACE2 cells against Omicron BA.1 strain). However, galactosidase inhibitors did not exhibit antiviral activity, whereas mannosidase inhibitors were both active and cytotoxic. As our iminosugar-based drug candidates act by a host-directed mechanism, they should be more resilient to drug resistance. Moreover, this strategy could be extended to identify potential drug candidates for other viral infections.
PB  - Taylor and Francis Group
T2  - Journal of Enzyme Inhibition and Medicinal Chemistry
T1  - Development of iminosugar-based glycosidase inhibitors as drug candidates for SARS-CoV-2 virus via molecular modelling and in vitro studies
VL  - 39
IS  - 1
SP  - 2289007
DO  - 10.1080/14756366.2023.2289007
ER  - 
@article{
author = "Ferjančić, Zorana and Bihelović, Filip and Vulović, Bojan and Matović, Radomir and Trmčić, Milena and Janković, Aleksandar and Pavlović, Miloš and Đurković, Filip T. and Prodanović, Radivoje and Đurđević Đelmaš, Aleksandra and Kaličanin, Nevena and Zlatović, Mario and Sladić, Dušan and Vallet, Thomas and Vignuzzi, Marco and Saičić, Radomir N.",
year = "2024",
abstract = "We developed new iminosugar-based glycosidase inhibitors against SARS-CoV-2. Known drugs (miglustat, migalastat, miglitol, and swainsonine) were chosen as lead compounds to develop three classes of glycosidase inhibitors (α-glucosidase, α-galactosidase, and mannosidase). Molecular modelling of the lead compounds, synthesis of the compounds with the highest docking scores, enzyme inhibition tests, and in vitro antiviral assays afforded rationally designed inhibitors. Two highly active α-glucosidase inhibitors were discovered, where one of them is the most potent iminosugar-based anti-SARS-CoV-2 agent to date (EC90 = 1.94 µM in A549-ACE2 cells against Omicron BA.1 strain). However, galactosidase inhibitors did not exhibit antiviral activity, whereas mannosidase inhibitors were both active and cytotoxic. As our iminosugar-based drug candidates act by a host-directed mechanism, they should be more resilient to drug resistance. Moreover, this strategy could be extended to identify potential drug candidates for other viral infections.",
publisher = "Taylor and Francis Group",
journal = "Journal of Enzyme Inhibition and Medicinal Chemistry",
title = "Development of iminosugar-based glycosidase inhibitors as drug candidates for SARS-CoV-2 virus via molecular modelling and in vitro studies",
volume = "39",
number = "1",
pages = "2289007",
doi = "10.1080/14756366.2023.2289007"
}
Ferjančić, Z., Bihelović, F., Vulović, B., Matović, R., Trmčić, M., Janković, A., Pavlović, M., Đurković, F. T., Prodanović, R., Đurđević Đelmaš, A., Kaličanin, N., Zlatović, M., Sladić, D., Vallet, T., Vignuzzi, M.,& Saičić, R. N.. (2024). Development of iminosugar-based glycosidase inhibitors as drug candidates for SARS-CoV-2 virus via molecular modelling and in vitro studies. in Journal of Enzyme Inhibition and Medicinal Chemistry
Taylor and Francis Group., 39(1), 2289007.
https://doi.org/10.1080/14756366.2023.2289007
Ferjančić Z, Bihelović F, Vulović B, Matović R, Trmčić M, Janković A, Pavlović M, Đurković FT, Prodanović R, Đurđević Đelmaš A, Kaličanin N, Zlatović M, Sladić D, Vallet T, Vignuzzi M, Saičić RN. Development of iminosugar-based glycosidase inhibitors as drug candidates for SARS-CoV-2 virus via molecular modelling and in vitro studies. in Journal of Enzyme Inhibition and Medicinal Chemistry. 2024;39(1):2289007.
doi:10.1080/14756366.2023.2289007 .
Ferjančić, Zorana, Bihelović, Filip, Vulović, Bojan, Matović, Radomir, Trmčić, Milena, Janković, Aleksandar, Pavlović, Miloš, Đurković, Filip T., Prodanović, Radivoje, Đurđević Đelmaš, Aleksandra, Kaličanin, Nevena, Zlatović, Mario, Sladić, Dušan, Vallet, Thomas, Vignuzzi, Marco, Saičić, Radomir N., "Development of iminosugar-based glycosidase inhibitors as drug candidates for SARS-CoV-2 virus via molecular modelling and in vitro studies" in Journal of Enzyme Inhibition and Medicinal Chemistry, 39, no. 1 (2024):2289007,
https://doi.org/10.1080/14756366.2023.2289007 . .
4
2
1

Gold(I)-Catalyzed Domino Cyclizations of Diynes for the Synthesis of Functionalized Cyclohexenone Derivatives. Total Synthesis of (-)-Gabosine H and (-)-6-epi-Gabosine H

Vulović, Bojan; Kolarski, Dusan; Bihelović, Filip; Matović, Radomir; Gruden, Maja; Saičić, Radomir N.

(American Chemical Society (ACS), 2016)

TY  - JOUR
AU  - Vulović, Bojan
AU  - Kolarski, Dusan
AU  - Bihelović, Filip
AU  - Matović, Radomir
AU  - Gruden, Maja
AU  - Saičić, Radomir N.
PY  - 2016
UR  - https://cer.ihtm.bg.ac.rs/handle/123456789/1847
AB  - 1,6-Diynes with a t-butylcarbonate group in the propargylic position undergo gold(I)-catalyzed dominocyclization which affords alpha-hydroxycyclohexenones. The described sequence can be applied on functionalized, highly oxygenated substrates, as examplified in the synthesis of (-)-gabosine H and its epimer.
PB  - American Chemical Society (ACS)
T2  - Organic Letters
T1  - Gold(I)-Catalyzed Domino Cyclizations of Diynes for the Synthesis of Functionalized Cyclohexenone Derivatives. Total Synthesis of (-)-Gabosine H and (-)-6-epi-Gabosine H
VL  - 18
IS  - 15
SP  - 3886
EP  - 3889
DO  - 10.1021/acs.orglett.6b01898
ER  - 
@article{
author = "Vulović, Bojan and Kolarski, Dusan and Bihelović, Filip and Matović, Radomir and Gruden, Maja and Saičić, Radomir N.",
year = "2016",
abstract = "1,6-Diynes with a t-butylcarbonate group in the propargylic position undergo gold(I)-catalyzed dominocyclization which affords alpha-hydroxycyclohexenones. The described sequence can be applied on functionalized, highly oxygenated substrates, as examplified in the synthesis of (-)-gabosine H and its epimer.",
publisher = "American Chemical Society (ACS)",
journal = "Organic Letters",
title = "Gold(I)-Catalyzed Domino Cyclizations of Diynes for the Synthesis of Functionalized Cyclohexenone Derivatives. Total Synthesis of (-)-Gabosine H and (-)-6-epi-Gabosine H",
volume = "18",
number = "15",
pages = "3886-3889",
doi = "10.1021/acs.orglett.6b01898"
}
Vulović, B., Kolarski, D., Bihelović, F., Matović, R., Gruden, M.,& Saičić, R. N.. (2016). Gold(I)-Catalyzed Domino Cyclizations of Diynes for the Synthesis of Functionalized Cyclohexenone Derivatives. Total Synthesis of (-)-Gabosine H and (-)-6-epi-Gabosine H. in Organic Letters
American Chemical Society (ACS)., 18(15), 3886-3889.
https://doi.org/10.1021/acs.orglett.6b01898
Vulović B, Kolarski D, Bihelović F, Matović R, Gruden M, Saičić RN. Gold(I)-Catalyzed Domino Cyclizations of Diynes for the Synthesis of Functionalized Cyclohexenone Derivatives. Total Synthesis of (-)-Gabosine H and (-)-6-epi-Gabosine H. in Organic Letters. 2016;18(15):3886-3889.
doi:10.1021/acs.orglett.6b01898 .
Vulović, Bojan, Kolarski, Dusan, Bihelović, Filip, Matović, Radomir, Gruden, Maja, Saičić, Radomir N., "Gold(I)-Catalyzed Domino Cyclizations of Diynes for the Synthesis of Functionalized Cyclohexenone Derivatives. Total Synthesis of (-)-Gabosine H and (-)-6-epi-Gabosine H" in Organic Letters, 18, no. 15 (2016):3886-3889,
https://doi.org/10.1021/acs.orglett.6b01898 . .
10
17
11
18

Synthesis of endoperoxides by domino reactions of ketones and molecular oxygen

Novkovic, L; Trmcic, M; Rodić, Marko V.; Bihelović, Filip; Zlatar, Matija; Matović, Radomir; Saičić, Radomir N.

(Royal Soc Chemistry, Cambridge, 2015)

TY  - JOUR
AU  - Novkovic, L
AU  - Trmcic, M
AU  - Rodić, Marko V.
AU  - Bihelović, Filip
AU  - Zlatar, Matija
AU  - Matović, Radomir
AU  - Saičić, Radomir N.
PY  - 2015
UR  - https://cer.ihtm.bg.ac.rs/handle/123456789/1796
AB  - Domino reactions of ketones with molecular oxygen in the presence of potassium hydroxide and potassium t-butoxide afford cyclic hydroperoxy acetals (3,5-dihydroxy-1,2-dioxanes). Mixed endoperoxides can also be obtained in a three-component reaction of two ketones and oxygen.
PB  - Royal Soc Chemistry, Cambridge
T2  - RSC Advances
T1  - Synthesis of endoperoxides by domino reactions of ketones and molecular oxygen
VL  - 5
IS  - 120
SP  - 99577
EP  - 99584
DO  - 10.1039/c5ra13476e
ER  - 
@article{
author = "Novkovic, L and Trmcic, M and Rodić, Marko V. and Bihelović, Filip and Zlatar, Matija and Matović, Radomir and Saičić, Radomir N.",
year = "2015",
abstract = "Domino reactions of ketones with molecular oxygen in the presence of potassium hydroxide and potassium t-butoxide afford cyclic hydroperoxy acetals (3,5-dihydroxy-1,2-dioxanes). Mixed endoperoxides can also be obtained in a three-component reaction of two ketones and oxygen.",
publisher = "Royal Soc Chemistry, Cambridge",
journal = "RSC Advances",
title = "Synthesis of endoperoxides by domino reactions of ketones and molecular oxygen",
volume = "5",
number = "120",
pages = "99577-99584",
doi = "10.1039/c5ra13476e"
}
Novkovic, L., Trmcic, M., Rodić, M. V., Bihelović, F., Zlatar, M., Matović, R.,& Saičić, R. N.. (2015). Synthesis of endoperoxides by domino reactions of ketones and molecular oxygen. in RSC Advances
Royal Soc Chemistry, Cambridge., 5(120), 99577-99584.
https://doi.org/10.1039/c5ra13476e
Novkovic L, Trmcic M, Rodić MV, Bihelović F, Zlatar M, Matović R, Saičić RN. Synthesis of endoperoxides by domino reactions of ketones and molecular oxygen. in RSC Advances. 2015;5(120):99577-99584.
doi:10.1039/c5ra13476e .
Novkovic, L, Trmcic, M, Rodić, Marko V., Bihelović, Filip, Zlatar, Matija, Matović, Radomir, Saičić, Radomir N., "Synthesis of endoperoxides by domino reactions of ketones and molecular oxygen" in RSC Advances, 5, no. 120 (2015):99577-99584,
https://doi.org/10.1039/c5ra13476e . .
10
6
9

Total synthesis and biological evaluation of atrop-O-benzyl-desmethylabyssomicin C

Matović, Radomir; Bihelović, Filip; Gruden-Pavlović, Maja; Saičić, Radomir N.

(Royal Soc Chemistry, Cambridge, 2014)

TY  - JOUR
AU  - Matović, Radomir
AU  - Bihelović, Filip
AU  - Gruden-Pavlović, Maja
AU  - Saičić, Radomir N.
PY  - 2014
UR  - https://cer.ihtm.bg.ac.rs/handle/123456789/1400
AB  - The total synthesis of desmethylabyssomicin C analogue 1 was accomplished using diastereotopos-selective ring closing metathesis and Nozaki-Hiyama-Kishi cyclization as the key steps. The synthetic analogue retained its antibacterial activity against methicillin-resistant S. aureus strains, whereas its cytotoxicity decreased for three orders of magnitude, as compared to atrop-abyssomicin C.
PB  - Royal Soc Chemistry, Cambridge
T2  - Organic & Biomolecular Chemistry
T1  - Total synthesis and biological evaluation of atrop-O-benzyl-desmethylabyssomicin C
VL  - 12
IS  - 39
SP  - 7682
EP  - 7685
DO  - 10.1039/c4ob01436g
ER  - 
@article{
author = "Matović, Radomir and Bihelović, Filip and Gruden-Pavlović, Maja and Saičić, Radomir N.",
year = "2014",
abstract = "The total synthesis of desmethylabyssomicin C analogue 1 was accomplished using diastereotopos-selective ring closing metathesis and Nozaki-Hiyama-Kishi cyclization as the key steps. The synthetic analogue retained its antibacterial activity against methicillin-resistant S. aureus strains, whereas its cytotoxicity decreased for three orders of magnitude, as compared to atrop-abyssomicin C.",
publisher = "Royal Soc Chemistry, Cambridge",
journal = "Organic & Biomolecular Chemistry",
title = "Total synthesis and biological evaluation of atrop-O-benzyl-desmethylabyssomicin C",
volume = "12",
number = "39",
pages = "7682-7685",
doi = "10.1039/c4ob01436g"
}
Matović, R., Bihelović, F., Gruden-Pavlović, M.,& Saičić, R. N.. (2014). Total synthesis and biological evaluation of atrop-O-benzyl-desmethylabyssomicin C. in Organic & Biomolecular Chemistry
Royal Soc Chemistry, Cambridge., 12(39), 7682-7685.
https://doi.org/10.1039/c4ob01436g
Matović R, Bihelović F, Gruden-Pavlović M, Saičić RN. Total synthesis and biological evaluation of atrop-O-benzyl-desmethylabyssomicin C. in Organic & Biomolecular Chemistry. 2014;12(39):7682-7685.
doi:10.1039/c4ob01436g .
Matović, Radomir, Bihelović, Filip, Gruden-Pavlović, Maja, Saičić, Radomir N., "Total synthesis and biological evaluation of atrop-O-benzyl-desmethylabyssomicin C" in Organic & Biomolecular Chemistry, 12, no. 39 (2014):7682-7685,
https://doi.org/10.1039/c4ob01436g . .
14
12
12

Diastereoselective addition of alkenylchromium(III) reagents to Garner's aldehyde. The Nozaki-Hiyama-Kishi coupling approach to sphingosines and ceramides

Ferjančić, Zorana; Matović, Radomir; Bihelović, Filip

(Serbian Chemical Soc, Belgrade, 2014)

TY  - JOUR
AU  - Ferjančić, Zorana
AU  - Matović, Radomir
AU  - Bihelović, Filip
PY  - 2014
UR  - https://cer.ihtm.bg.ac.rs/handle/123456789/1557
AB  - Intermolecular Nozaki-Hiyama-Kishi coupling between alkenylchromium(III) reagents, derived from either (E)-(2-bromoethenyl)benzene or (E)-1-iodo-1-pentadecene, and the conformationally rigid Garner's aldehyde resulted in the stereoselective formation of Felkin-type allylic alcohols in good yields, thus providing an easy access to sphingosines. In addition, when the protecting group in the Garner's aldehyde was changed (from Boc to N-octanoyl), a reversal of stereoselectivity was observed in the reaction with (E)-1-pentadecenylchromium(III), probably as the result of hydrophobic interactions between the long carbon chains of the reaction partners.
PB  - Serbian Chemical Soc, Belgrade
T2  - Journal of the Serbian Chemical Society
T1  - Diastereoselective addition of alkenylchromium(III) reagents to Garner's aldehyde. The Nozaki-Hiyama-Kishi coupling approach to sphingosines and ceramides
VL  - 79
IS  - 6
SP  - 627
EP  - 636
DO  - 10.2298/JSC130611067F
ER  - 
@article{
author = "Ferjančić, Zorana and Matović, Radomir and Bihelović, Filip",
year = "2014",
abstract = "Intermolecular Nozaki-Hiyama-Kishi coupling between alkenylchromium(III) reagents, derived from either (E)-(2-bromoethenyl)benzene or (E)-1-iodo-1-pentadecene, and the conformationally rigid Garner's aldehyde resulted in the stereoselective formation of Felkin-type allylic alcohols in good yields, thus providing an easy access to sphingosines. In addition, when the protecting group in the Garner's aldehyde was changed (from Boc to N-octanoyl), a reversal of stereoselectivity was observed in the reaction with (E)-1-pentadecenylchromium(III), probably as the result of hydrophobic interactions between the long carbon chains of the reaction partners.",
publisher = "Serbian Chemical Soc, Belgrade",
journal = "Journal of the Serbian Chemical Society",
title = "Diastereoselective addition of alkenylchromium(III) reagents to Garner's aldehyde. The Nozaki-Hiyama-Kishi coupling approach to sphingosines and ceramides",
volume = "79",
number = "6",
pages = "627-636",
doi = "10.2298/JSC130611067F"
}
Ferjančić, Z., Matović, R.,& Bihelović, F.. (2014). Diastereoselective addition of alkenylchromium(III) reagents to Garner's aldehyde. The Nozaki-Hiyama-Kishi coupling approach to sphingosines and ceramides. in Journal of the Serbian Chemical Society
Serbian Chemical Soc, Belgrade., 79(6), 627-636.
https://doi.org/10.2298/JSC130611067F
Ferjančić Z, Matović R, Bihelović F. Diastereoselective addition of alkenylchromium(III) reagents to Garner's aldehyde. The Nozaki-Hiyama-Kishi coupling approach to sphingosines and ceramides. in Journal of the Serbian Chemical Society. 2014;79(6):627-636.
doi:10.2298/JSC130611067F .
Ferjančić, Zorana, Matović, Radomir, Bihelović, Filip, "Diastereoselective addition of alkenylchromium(III) reagents to Garner's aldehyde. The Nozaki-Hiyama-Kishi coupling approach to sphingosines and ceramides" in Journal of the Serbian Chemical Society, 79, no. 6 (2014):627-636,
https://doi.org/10.2298/JSC130611067F . .
2
2
2

Total synthesis and biological evaluation of (-)-atrop-abyssomicin C

Bihelović, Filip; Karadžić, Ivanka; Matović, Radomir; Saičić, Radomir N.

(Royal Soc Chemistry, Cambridge, 2013)

TY  - JOUR
AU  - Bihelović, Filip
AU  - Karadžić, Ivanka
AU  - Matović, Radomir
AU  - Saičić, Radomir N.
PY  - 2013
UR  - https://cer.ihtm.bg.ac.rs/handle/123456789/1214
AB  - Enantioselective synthesis of a marine antibiotic (-)-atrop-abyssomicin C was accomplished in 21 steps, in 1.8% overall yield (4%, based on the recovered starting material). The key steps of the synthesis are the formation of the functionalized cyclohexane core by an organocatalyzed Tsuji-Trost reaction, the formation of a tricyclic spirotetronate unit by a gold-catalyzed reaction sequence and the highly efficient eleven-membered ring closure by a Nozaki-Hiyama-Kishi reaction. Biological tests showed all abyssomicin derivatives to possess strong antibacterial activity against methicillin resistant S. aureus strains; however, they also proved to be cytotoxic, both to malignant and to normal somatic cells.
PB  - Royal Soc Chemistry, Cambridge
T2  - Organic & Biomolecular Chemistry
T1  - Total synthesis and biological evaluation of (-)-atrop-abyssomicin C
VL  - 11
IS  - 33
SP  - 5413
EP  - 5424
DO  - 10.1039/c3ob40692j
ER  - 
@article{
author = "Bihelović, Filip and Karadžić, Ivanka and Matović, Radomir and Saičić, Radomir N.",
year = "2013",
abstract = "Enantioselective synthesis of a marine antibiotic (-)-atrop-abyssomicin C was accomplished in 21 steps, in 1.8% overall yield (4%, based on the recovered starting material). The key steps of the synthesis are the formation of the functionalized cyclohexane core by an organocatalyzed Tsuji-Trost reaction, the formation of a tricyclic spirotetronate unit by a gold-catalyzed reaction sequence and the highly efficient eleven-membered ring closure by a Nozaki-Hiyama-Kishi reaction. Biological tests showed all abyssomicin derivatives to possess strong antibacterial activity against methicillin resistant S. aureus strains; however, they also proved to be cytotoxic, both to malignant and to normal somatic cells.",
publisher = "Royal Soc Chemistry, Cambridge",
journal = "Organic & Biomolecular Chemistry",
title = "Total synthesis and biological evaluation of (-)-atrop-abyssomicin C",
volume = "11",
number = "33",
pages = "5413-5424",
doi = "10.1039/c3ob40692j"
}
Bihelović, F., Karadžić, I., Matović, R.,& Saičić, R. N.. (2013). Total synthesis and biological evaluation of (-)-atrop-abyssomicin C. in Organic & Biomolecular Chemistry
Royal Soc Chemistry, Cambridge., 11(33), 5413-5424.
https://doi.org/10.1039/c3ob40692j
Bihelović F, Karadžić I, Matović R, Saičić RN. Total synthesis and biological evaluation of (-)-atrop-abyssomicin C. in Organic & Biomolecular Chemistry. 2013;11(33):5413-5424.
doi:10.1039/c3ob40692j .
Bihelović, Filip, Karadžić, Ivanka, Matović, Radomir, Saičić, Radomir N., "Total synthesis and biological evaluation of (-)-atrop-abyssomicin C" in Organic & Biomolecular Chemistry, 11, no. 33 (2013):5413-5424,
https://doi.org/10.1039/c3ob40692j . .
1
29
26
28

Corrigendum to: Organocatalyzed Tsuji-Trost reaction: a new method for the closure of five- and six-membered rings (vol 65, pg 10485, 2009)

Vulović, Bojan; Bihelović, Filip; Matović, Radomir; Saičić, Radomir N.

(Oxford : Pergamon-Elsevier Science Ltd, 2010)

TY  - JOUR
AU  - Vulović, Bojan
AU  - Bihelović, Filip
AU  - Matović, Radomir
AU  - Saičić, Radomir N.
PY  - 2010
UR  - https://cer.ihtm.bg.ac.rs/handle/123456789/658
PB  - Oxford : Pergamon-Elsevier Science Ltd
T2  - Tetrahedron
T1  - Corrigendum to: Organocatalyzed Tsuji-Trost reaction: a new method for the closure of five- and six-membered rings (vol 65, pg 10485, 2009)
VL  - 66
IS  - 17
SP  - 3275
EP  - 3275
DO  - 10.1016/j.tet.2010.03.013
ER  - 
@article{
author = "Vulović, Bojan and Bihelović, Filip and Matović, Radomir and Saičić, Radomir N.",
year = "2010",
publisher = "Oxford : Pergamon-Elsevier Science Ltd",
journal = "Tetrahedron",
title = "Corrigendum to: Organocatalyzed Tsuji-Trost reaction: a new method for the closure of five- and six-membered rings (vol 65, pg 10485, 2009)",
volume = "66",
number = "17",
pages = "3275-3275",
doi = "10.1016/j.tet.2010.03.013"
}
Vulović, B., Bihelović, F., Matović, R.,& Saičić, R. N.. (2010). Corrigendum to: Organocatalyzed Tsuji-Trost reaction: a new method for the closure of five- and six-membered rings (vol 65, pg 10485, 2009). in Tetrahedron
Oxford : Pergamon-Elsevier Science Ltd., 66(17), 3275-3275.
https://doi.org/10.1016/j.tet.2010.03.013
Vulović B, Bihelović F, Matović R, Saičić RN. Corrigendum to: Organocatalyzed Tsuji-Trost reaction: a new method for the closure of five- and six-membered rings (vol 65, pg 10485, 2009). in Tetrahedron. 2010;66(17):3275-3275.
doi:10.1016/j.tet.2010.03.013 .
Vulović, Bojan, Bihelović, Filip, Matović, Radomir, Saičić, Radomir N., "Corrigendum to: Organocatalyzed Tsuji-Trost reaction: a new method for the closure of five- and six-membered rings (vol 65, pg 10485, 2009)" in Tetrahedron, 66, no. 17 (2010):3275-3275,
https://doi.org/10.1016/j.tet.2010.03.013 . .
4
7
3

Organocatalyzed Tsuji-Trost reaction: a new method for the closure of five- and six-membered rings

Vulović, Bojan; Bihelović, Filip; Matović, Radomir; Saičić, Radomir N.

(Oxford : Pergamon-Elsevier Science Ltd, 2009)

TY  - JOUR
AU  - Vulović, Bojan
AU  - Bihelović, Filip
AU  - Matović, Radomir
AU  - Saičić, Radomir N.
PY  - 2009
UR  - http://cherry.chem.bg.ac.rs/handle/123456789/1031
UR  - https://cer.ihtm.bg.ac.rs/handle/123456789/2774
AB  - A combination of organotransition metal catalysis and organocatalysis allows for Tsuji-Trost 5-exo- and 6-exo-cyclizations of aldehydes. This transformation can also be accomplished as a catalytic asymmetric reaction, which affords vinylcyclopentane derivatives with up to 98%ee. (C) 2009 Elsevier Ltd. All rights reserved.
PB  - Oxford : Pergamon-Elsevier Science Ltd
T2  - Tetrahedron
T1  - Organocatalyzed Tsuji-Trost reaction: a new method for the closure of five- and six-membered rings
VL  - 65
IS  - 50
SP  - 10485
EP  - 10494
DO  - 10.1016/j.tet.2009.10.006
ER  - 
@article{
author = "Vulović, Bojan and Bihelović, Filip and Matović, Radomir and Saičić, Radomir N.",
year = "2009",
abstract = "A combination of organotransition metal catalysis and organocatalysis allows for Tsuji-Trost 5-exo- and 6-exo-cyclizations of aldehydes. This transformation can also be accomplished as a catalytic asymmetric reaction, which affords vinylcyclopentane derivatives with up to 98%ee. (C) 2009 Elsevier Ltd. All rights reserved.",
publisher = "Oxford : Pergamon-Elsevier Science Ltd",
journal = "Tetrahedron",
title = "Organocatalyzed Tsuji-Trost reaction: a new method for the closure of five- and six-membered rings",
volume = "65",
number = "50",
pages = "10485-10494",
doi = "10.1016/j.tet.2009.10.006"
}
Vulović, B., Bihelović, F., Matović, R.,& Saičić, R. N.. (2009). Organocatalyzed Tsuji-Trost reaction: a new method for the closure of five- and six-membered rings. in Tetrahedron
Oxford : Pergamon-Elsevier Science Ltd., 65(50), 10485-10494.
https://doi.org/10.1016/j.tet.2009.10.006
Vulović B, Bihelović F, Matović R, Saičić RN. Organocatalyzed Tsuji-Trost reaction: a new method for the closure of five- and six-membered rings. in Tetrahedron. 2009;65(50):10485-10494.
doi:10.1016/j.tet.2009.10.006 .
Vulović, Bojan, Bihelović, Filip, Matović, Radomir, Saičić, Radomir N., "Organocatalyzed Tsuji-Trost reaction: a new method for the closure of five- and six-membered rings" in Tetrahedron, 65, no. 50 (2009):10485-10494,
https://doi.org/10.1016/j.tet.2009.10.006 . .
65
44
61

Organocatalyzed cyclizations of π-allylpalladium complexes: A new method for the construction of five- and six-membered rings

Bihelović, Filip; Matović, Radomir; Vulović, Bojan; Saičić, Radomir N.

(American Chemical Society (ACS), 2007)

TY  - JOUR
AU  - Bihelović, Filip
AU  - Matović, Radomir
AU  - Vulović, Bojan
AU  - Saičić, Radomir N.
PY  - 2007
UR  - https://cer.ihtm.bg.ac.rs/handle/123456789/343
AB  - Synergic combination of organotransition metal catalysis and organocatalysis allows, for the first time, the Tsuji-Trost cyclization of aldehydes. A catalytic asymmetric variant of the reaction is also possible.
PB  - American Chemical Society (ACS)
T2  - Organic Letters
T1  - Organocatalyzed cyclizations of π-allylpalladium complexes: A new method for the construction of five- and six-membered rings
VL  - 9
IS  - 24
SP  - 5063
EP  - 5066
DO  - 10.1021/ol7023554
ER  - 
@article{
author = "Bihelović, Filip and Matović, Radomir and Vulović, Bojan and Saičić, Radomir N.",
year = "2007",
abstract = "Synergic combination of organotransition metal catalysis and organocatalysis allows, for the first time, the Tsuji-Trost cyclization of aldehydes. A catalytic asymmetric variant of the reaction is also possible.",
publisher = "American Chemical Society (ACS)",
journal = "Organic Letters",
title = "Organocatalyzed cyclizations of π-allylpalladium complexes: A new method for the construction of five- and six-membered rings",
volume = "9",
number = "24",
pages = "5063-5066",
doi = "10.1021/ol7023554"
}
Bihelović, F., Matović, R., Vulović, B.,& Saičić, R. N.. (2007). Organocatalyzed cyclizations of π-allylpalladium complexes: A new method for the construction of five- and six-membered rings. in Organic Letters
American Chemical Society (ACS)., 9(24), 5063-5066.
https://doi.org/10.1021/ol7023554
Bihelović F, Matović R, Vulović B, Saičić RN. Organocatalyzed cyclizations of π-allylpalladium complexes: A new method for the construction of five- and six-membered rings. in Organic Letters. 2007;9(24):5063-5066.
doi:10.1021/ol7023554 .
Bihelović, Filip, Matović, Radomir, Vulović, Bojan, Saičić, Radomir N., "Organocatalyzed cyclizations of π-allylpalladium complexes: A new method for the construction of five- and six-membered rings" in Organic Letters, 9, no. 24 (2007):5063-5066,
https://doi.org/10.1021/ol7023554 . .
120
96
108

Erratum: Organocatalyzed Cyclizations of pi-allylpalladium complexes: A new method for the construction of five- and six-membered rings (vol 9, pg 5064, 2007)

Bihelović, Filip; Matović, Radomir; Vulović, Bojan; Saičić, Radomir N.

(American Chemical Society (ACS), 2007)

TY  - JOUR
AU  - Bihelović, Filip
AU  - Matović, Radomir
AU  - Vulović, Bojan
AU  - Saičić, Radomir N.
PY  - 2007
UR  - http://cherry.chem.bg.ac.rs/handle/123456789/894
UR  - https://cer.ihtm.bg.ac.rs/handle/123456789/2773
AB  - Page 5064. Two references pertinent to the described work have been omitted in ref 13:  For the first example of combining organocatalysis and transition metal catalysis, see:  (e) Jellerichs, B. G.; Kong, J.-R.; Krische, M. J. J. Am. Chem. Soc. 2003, 125, 7758. For a recent application of double catalysis to a highly efficient asymmetric allylation of aldehydes, see:  (f) Mukherjee, S.; List, B. J. Am. Chem. Soc. 2007, 129, 11336.11/28/2007
PB  - American Chemical Society (ACS)
T2  - Organic Letters
T1  - Erratum: Organocatalyzed Cyclizations of pi-allylpalladium complexes: A new method for the construction of five- and six-membered rings (vol 9, pg 5064, 2007)
VL  - 9
IS  - 26
SP  - 5649
EP  - 5649
DO  - 10.1021/ol702760g
ER  - 
@article{
author = "Bihelović, Filip and Matović, Radomir and Vulović, Bojan and Saičić, Radomir N.",
year = "2007",
abstract = "Page 5064. Two references pertinent to the described work have been omitted in ref 13:  For the first example of combining organocatalysis and transition metal catalysis, see:  (e) Jellerichs, B. G.; Kong, J.-R.; Krische, M. J. J. Am. Chem. Soc. 2003, 125, 7758. For a recent application of double catalysis to a highly efficient asymmetric allylation of aldehydes, see:  (f) Mukherjee, S.; List, B. J. Am. Chem. Soc. 2007, 129, 11336.11/28/2007",
publisher = "American Chemical Society (ACS)",
journal = "Organic Letters",
title = "Erratum: Organocatalyzed Cyclizations of pi-allylpalladium complexes: A new method for the construction of five- and six-membered rings (vol 9, pg 5064, 2007)",
volume = "9",
number = "26",
pages = "5649-5649",
doi = "10.1021/ol702760g"
}
Bihelović, F., Matović, R., Vulović, B.,& Saičić, R. N.. (2007). Erratum: Organocatalyzed Cyclizations of pi-allylpalladium complexes: A new method for the construction of five- and six-membered rings (vol 9, pg 5064, 2007). in Organic Letters
American Chemical Society (ACS)., 9(26), 5649-5649.
https://doi.org/10.1021/ol702760g
Bihelović F, Matović R, Vulović B, Saičić RN. Erratum: Organocatalyzed Cyclizations of pi-allylpalladium complexes: A new method for the construction of five- and six-membered rings (vol 9, pg 5064, 2007). in Organic Letters. 2007;9(26):5649-5649.
doi:10.1021/ol702760g .
Bihelović, Filip, Matović, Radomir, Vulović, Bojan, Saičić, Radomir N., "Erratum: Organocatalyzed Cyclizations of pi-allylpalladium complexes: A new method for the construction of five- and six-membered rings (vol 9, pg 5064, 2007)" in Organic Letters, 9, no. 26 (2007):5649-5649,
https://doi.org/10.1021/ol702760g . .
4
3
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