Претраживање
Приказ резултата 31-40 од 300
A refined pharmacophore identifies potent 4-amino-7-chloroquinoline-based inhibitors of the botulinum neurotoxin serotype A metalloprotease
(American Chemical Society (ACS), 2007)
We previously identified structurally diverse small molecule (non-peptidic) inhibitors (SMNPIs) of the botulinum neurotoxin serotype A (BoNT/A) light chain (LC). Of these, several (including antimalarial drugs) contained ...
Determination of glass temperature of polymers by inverse gas chromatography
(Elsevier, 2008)
Inverse gas chromatography (IGC) is an attractive technique for polymer characterization due to possible simultaneous determination of various physicochemical properties of polymer systems merely from retention times of ...
Novel 4-aminoquinolines active against chloroquine-resistant and sensitive P. falciparum strains that also inhibit botulinum serotype A
(American Chemical Society (ACS), 2008)
We report on the initial result of the coupling of 4-amino-7- chloroquinoline with steroidal and adamantane constituents to provide small molecules with excellent in vitro antimalarial activities (IC90 (W2) down to 6.74 ...
New chimeric antimalarials with 4-aminoquinoline moiety linked to a tetraoxane skeleton
(American Chemical Society (ACS), 2008)
The synthesis of the chimeric molecules consisting of two pharmacophores, tetraoxane and 7-chloro-4-aminoquinoline, is reported. The tetraoxanes 2, 4, and 8 show relatively potent in vitro antimalarial activities, with ...
Synthesis and antioxidant properties of fullero-steroidal covalent conjugates
(Oxford : Pergamon-Elsevier Science Ltd, 2007)
Four new fullero-steroids were synthesized starting from gamma-aminobutyric acid (GABA)-incorporated fulleropyrrolidine and corresponding sterols. The synthesis, characterization, preliminary study on in vitro antioxidant ...
Influence of thermal treatment on phenolic compounds and antioxidant properties of oak acorns from Serbia
(Elsevier, 2007)
The aim of the present work was to investigate and compare phenolic compounds and antioxidant activity of methanol extracts of Quercus robur and Quercus cerris acorn kernels obtained before and after thermal treatment. ...
Fluctuations of the number of particles and mass adsorbed on the sensor surface surrounded by a mixture of an arbitrary number of gases
(Elsevier, 2007)
In this paper the theory of the adsorption and desorption process of an arbitrary number of gases on the sensor surface is presented. It is assumed that the sorption follows the Langmuir isotherm. The exact expressions are ...
Coordinating Benzenes Stack Stronger than Noncoordinating Benzenes, even at Large Horizontal Displacements
(American Chemical Society (ACS), 2016)
Stacking interactions between two benzene molecules that coordinate transition metal ions within organometallic sandwich and half-sandwich compounds were investigated by performing Cambridge Structural Database (CSD) search ...
Understanding the Effect of Energy Density and Formulation Factors on the Printability and Characteristics of SLS Irbesartan Tablets-Application of the Decision Tree Model
(MDPI, 2021)
Selective laser sintering (SLS) is a rapid prototyping technique for the production of three-dimensional objects through selectively sintering powder-based layer materials. The aim of the study was to investigate the effect ...
Photodegradation of thiacloprid using Fe/TiO2 as a heterogeneous photo-Fenton catalyst
(Elsevier, 2011)
Three Fe/TiO2 photocatalysts with different content of Fe (1.9, 7.2 and 13.9%, w/w) were synthesized by a simple deposition-precipitation method and characterized by XRD, SEM, N-2 physisorption at 77K and Mossbauer ...