Претраживање
Приказ резултата 41-50 од 557
1,2,3,4-Tetrahydroisoquinoline Derivatives as a Novel Deoxyribonuclease I Inhibitors
(Wiley, 2021)
Herein we report an assessment of 24 1,2,3,4-tetrahydroisoquinoline derivatives for potential DNase I (deoxyribonuclease I) inhibitory properties in vitro. Four of them inhibited DNase I with IC50 values below 200 μM. The ...
Polycyclic aromatic hydrocarbons and their relationship to maturity and paleoenvironmental settings in lacustrine sediments of the Neogene Toplica Basin, Serbia
(Switzerland : Springer Nature, 2021)
The study investigated the influence of maturity, biomass type, and depositional settings on the distribution and relative abundance of polycyclic aromatic hydrocarbons (PAHs) for lacustrine sediments collected from depths ...
How aromatic system size affects the sensitivities of highly energetic molecules?
(Royal Society of Chemistry, 2021)
Positive values of electrostatic potentials above the central regions of the molecular surface are strongly related to the high sensitivities of highly energetic molecules. The influence of aromatic system size on the ...
Structural and thermal properties of Sn–Ag alloys
(Elsevier, 2021)
Microstructure and thermal properties of slowly cooled Sn–10% Ag and Sn–20% Ag alloys were experimentally investigated in this study. It was found that microstructure of the studied alloys is composed of large, plate-like ...
On Multiple-Resonator-based Implementation of IEC/IEEE Standard P-Class Compliant PMUs
(MDPI, 2021)
This article deals with the implementation of the P-Class PMU compliant with IEC/IEEE
Standard 60255-118-1:2018 by usage of a multiple-resonator (MR)-based approach for harmonic
analysis having been proposed recently. ...
3D-QSAR, molecular docking and in silico ADMET studies of propiophenone derivatives with anti-HIV-1 protease activity
(Springer Nature, 2021)
HIV protease inhibitors are one of the most important agents for the treatment of HIV infection. In this work, molecular modeling studies combining 3D-QSAR, molecular docking, MESP, HOMO, and LUMO energy calculations were ...
Synthesis, characterization, antimicrobial and cytotoxic activity and DNA-binding properties of d-metal complexes with hydrazones of Girard’s T and P reagents
(Springer Science and Business Media Deutschland GmbH, 2021)
In this work synthesis, characterization and crystal structures of 1, Zn(II) complex ([ZnL1(NCS)2]), with (E)-1-(2-oxo-2-(2-(quinolin-2-ylmethylene)hydrazinyl)ethyl)pyridin-1-ium chloride (HL1Cl) and 2, Bi(III) complex ...
In vitro evaluation of antiproliferative properties of novel organotin(IV) carboxylate compounds with propanoic acid derivatives on a panel of human cancer cell lines
(MDPI, 2021)
The synthesis of novel triphenyltin(IV) compounds, Ph3SnLn (n = 1–3), with oxaprozin (3-(4,5-diphenyloxazol-2-yl)propanoic acid), HL1, and the new propanoic acid derivatives 3-(4,5bis(4-methoxylphenyl)oxazol-2-yl)propanoic ...
Toxicity investigation of CeO2 nanoparticles coated with glucose and exopolysaccharides levan and pullulan on the bacterium Vibrio fischeri and aquatic organisms Daphnia magna and Danio rerio
(Elsevier, 2021)
Cerium oxide nanoparticles (nCeO2) have widespread applications, but they can be hazardous to the environment. Some reports indicate the toxic effect of nCeO2 on tested animals, but literature data are mainly contradictory. ...
Application of machine-learning algorithms for better understanding of tableting properties of lactose co-processed with lipid excipients
(MDPI, 2021)
Co-processing (CP) provides superior properties to excipients and has become a reliable option to facilitated formulation and manufacturing of variety of solid dosage forms. Development of directly compressible formulations ...